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The mean elimination half-life (T-?) values for naltrexone and 6-?-naltrexol are 4 hours and 13 hours, respectively. Naltrexone and 6-?-naltrexol are dose proportional in terms of AUC and Cmax over the range of 50 to 200 mg and do not accumulate after 100 mg daily doses.
You should tell your doctor if any of the following side effects become severe or don’t go away: Nausea, vomiting, diarrhea, or constipation. Stomach pain or cramping. Loss of appetite. Headache. Dizziness. Nervousness, irritability, or anxiety. Tearfulness. Increased or decreased energy.
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