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The mean elimination half-life (T-?) values for naltrexone and 6-?-naltrexol are 4 hours and 13 hours, respectively. Naltrexone and 6-?-naltrexol are dose proportional in terms of AUC and Cmax over the range of 50 to 200 mg and do not accumulate after 100 mg daily doses.
No, you cannot get high on naltrexone. In fact, naltrexone is prescribed to treat opiate/opioid addiction and alcoholism by blocking the pleasurable and euphoric effects of these substances. It works by binding to opioid receptors in the central nervous system that these drugs normally occupy.
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The mean elimination half-life (T-?) values for naltrexone and 6-?-naltrexol are 4 hours and 13 hours, respectively. Naltrexone and 6-?-naltrexol are dose proportional in terms of AUC and Cmax over the range of 50 to 200 mg and do not accumulate after 100 mg daily doses.
No, you cannot get high on naltrexone. In fact, naltrexone is prescribed to treat opiate/opioid addiction and alcoholism by blocking the pleasurable and euphoric effects of these substances. It works by binding to opioid receptors in the central nervous system that these drugs normally occupy.
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